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Drug discovery
Simulations of Promising Indolizidine—
α
6-
β
2 Nicotinic Acetylcholine Receptor Complexes
Article
Year: 2021
Pages: 1
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Systematic Roadmap for Cancer Drug Screening Using Zebrafish Embryo Xenograft Cancer Models: Melanoma Cell Line as a Case Study
Article
Year: 2021
Pages: 1
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DeepR2cov: deep representation learning on heterogeneous drug networks to discover anti-inflammatory agents for COVID-19
Article
Year: 2021
Pages: 1
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Comment on: Targeting the HGF/c-MET pathway in advanced pancreatic cancer: a key element of treatment that limits primary tumour growth and eliminates metastasis
Article
Year: 2020
Pages: 2
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High-Throughput Approaches for the Identification of
Pseudomonas aeruginosa
Antivirulents
Article
Pages: 1
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Title: “Labels Matter: Is it stress or is it Trauma?”
Article
Year: 2021
Pages: 1
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Compound NSC84167 selectively targets NRF2-activated pancreatic cancer by inhibiting asparagine synthesis pathway
Article
Year: 2021
Pages: 1
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Drug discovery oncology in a mouse: concepts, models and limitations
Article
Pages: 1
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Meta-regression of randomized control trials with antithrombotics: weak correlation between net clinical benefit and all cause-mortality
Article
Year: 2021
Pages: 1
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Peptide VSAK maintains tissue glucose uptake and attenuates pro-inflammatory responses caused by LPS in an experimental model of the systemic inflammatory response syndrome: a PET study
Article
Year: 2021
Pages: 1
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High-throughput compound screening identifies navitoclax combined with irradiation as a candidate therapy for HPV-negative head and neck squamous cell carcinoma
Article
Year: 2021
Pages: 1
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A novel inhibitor L755507 efficiently blocks c-Myc–MAX heterodimerization and induces apoptosis in cancer cells
Article
Year: 2021
Pages: 1
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Anticancer effects of the combined Thai noni juice ethanolic extracts and 5-fluorouracil against cholangiocarcinoma cells in vitro and in vivo
Article
Year: 2021
Pages: 1
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Targeted delivery of cytotoxic proteins to prostate cancer via conjugation to small molecule urea-based PSMA inhibitors
Article
Year: 2021
Pages: 1
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PAX8 lineage-driven T cell engaging antibody for the treatment of high-grade serous ovarian cancer
Article
Year: 2021
Pages: 1
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VALD-3, a Schiff base ligand synthesized from o-vanillin derivatives, induces cell cycle arrest and apoptosis in breast cancer cells by inhibiting the Wnt/β-catenin pathway
Article
Year: 2021
Pages: 1
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A Fine-Tuned Lipophilicity/Hydrophilicity Ratio Governs Antibacterial Potency and Selectivity of Bifurcated Halogen Bond-Forming NBTIs
Article
Year: 2021
Pages: 1
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Bacterial Natural Product Drug Discovery for New Antibiotics: Strategies for Tackling the Problem of Antibiotic Resistance by Efficient Bioprospecting
Article
Year: 2021
Pages: 1
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Acoustilytix™: A Web-Based Automated Ultrasonic Vocalization Scoring Platform
Article
Year: 2021
Pages: 1
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Identification of Potential Kinase Inhibitors within the PI3K/AKT Pathway of
Leishmania
Species
Article
Year: 2021
Pages: 1
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Discovery of Novel Allosteric Modulators Targeting an Extra-Helical Binding Site of GLP-1R Using Structure- and Ligand-Based Virtual Screening
Article
Year: 2021
Pages: 1
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Riminophenazine Derivatives as Potential Antituberculosis Agents: Synthesis, Biological, and Electrochemical Evaluations
Article
Year: 2021
Pages: 1
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Mycopharmaceuticals and Nutraceuticals: Promising Agents to Improve Human Well-Being and Life Quality
Article
Year: 2021
Pages: 1
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Transcriptome Profile Analysis of Triple-Negative Breast Cancer Cells in Response to a Novel Cytostatic Tetrahydroisoquinoline Compared to Paclitaxel
Article
Year: 2021
Pages: 1
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Metabolomic Characterization of a cf.
Neolyngbya
Cyanobacterium from the South China Sea Reveals Wenchangamide A, a Lipopeptide with In Vitro Apoptotic Potential in Colon Cancer Cells
Article
Year: 2021
Pages: 1
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Identification and Characterization of Novel Proteins from Arizona Bark Scorpion Venom That Inhibit Nav1.8, a Voltage-Gated Sodium Channel Regulator of Pain Signaling
Article
Year: 2021
Pages: 1
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Dopamine-loaded nanoparticle systems circumvent the blood–brain barrier restoring motor function in mouse model for Parkinson’s Disease
Article
Year: 2021
Pages: 1
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S494 O-glycosylation site on the SARS-CoV-2 RBD affects the virus affinity to ACE2 and its infectivity; a molecular dynamics study
Article
Year: 2021
Pages: 1
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N6-methyladenosine methyltransferases: functions, regulation, and clinical potential
Article
Year: 2021
Pages: 1
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Super enhancer regulation of cytokine-induced chemokine production in alcoholic hepatitis
Article
Year: 2021
Pages: 1
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Advances of Zebrafish in Neurodegenerative Disease: From Models to Drug Discovery
Article
Year: 2021
Pages: 1
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Abbreviated Profile of Drugs (APOD): modeling drug safety profiles to prioritize investigational COVID-19 treatments
Article
Year: 2021
Pages: 1
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Structure-guided microbial targeting of antistaphylococcal prodrugs
Article
Pages: 1
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A phenotypic high-content, high-throughput screen identifies inhibitors of NLRP3 inflammasome activation
Article
Year: 2021
Pages: 1
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Combining Genome-Wide Gene Expression Analysis (RNA-seq) and a Gene Editing Platform (CRISPR-Cas9) to Uncover the Selectively Pro-oxidant Activity of Aurone Compounds Against
Candida albicans
Article
Year: 2021
Pages: 1
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Comprehensive virtual screening of 4.8 k flavonoids reveals novel insights into allosteric inhibition of SARS-CoV-2 M
PRO
Article
Year: 2021
Pages: 1
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Designing a multi-epitope vaccine candidate to combat MERS-CoV by employing an immunoinformatics approach
Article
Year: 2021
Pages: 1
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Development of a CNS-permeable reactivator for nerve agent exposure: an iterative, multi-disciplinary approach
Article
Year: 2021
Pages: 1
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A phenomics approach for antiviral drug discovery
Article
Year: 2021
Pages: 1
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SARS-CoV-2-derived fusion inhibitor lipopeptides exhibit highly potent and broad-spectrum activity against divergent human coronaviruses
Article
Year: 2021
Pages: 1
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Plant Natural Flavonoids Against Multidrug Resistant Pathogens
Article
Year: 2021
Pages: 1
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Acetylation turns leucine into a drug by membrane transporter switching
Article
Year: 2021
Pages: 1
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Minimal mitochondrial respiration is required to prevent cell death by inhibition of mTOR signaling in CoQ-deficient cells
Article
Year: 2021
Pages: 1
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A proteomic platform to identify off-target proteins associated with therapeutic modalities that induce protein degradation or gene silencing
Article
Year: 2021
Pages: 1
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Conformational dynamics of androgen receptors bound to agonists and antagonists
Article
Year: 2021
Pages: 1
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Using Plate-Wash PCR and High-Throughput Sequencing to Measure Cultivated Diversity for Natural Product Discovery Efforts
Article
Year: 2021
Pages: 1
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A Novel Dialkylamino-Functionalized Chalcone, DML6, Inhibits Cervical Cancer Cell Proliferation, In Vitro, via Induction of Oxidative Stress, Intrinsic Apoptosis and Mitotic Catastrophe
Article
Year: 2021
Pages: 1
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Intranasal plus subcutaneous prime vaccination with a dual antigen COVID-19 vaccine elicits T-cell and antibody responses in mice
Article
Year: 2021
Pages: 1
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Real-world evidence for improved outcomes with histamine antagonists and aspirin in 22,560 COVID-19 patients
Article
Year: 2021
Pages: 1
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Defense of COVID-19 by Human Organoids
Article
Year: 2021
Pages: 16
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Anthelmintic resistance and homeostatic plasticity (
Brugia malayi
)
Article
Year: 2021
Pages: 1
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RETRACTED ARTICLE: Molecular detection of pathogenic
Escherichia coli
strains and their antibiogram associated with risk factors from diarrheic calves in Jimma Ethiopia
Article
Year: 2021
Pages: 1
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Traditional Chinese Medicine and Colorectal Cancer: Implications for Drug Discovery
Article
Year: 2021
Pages: 1
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Protective effects and mechanisms of high-dose vitamin C on sepsis-associated cognitive impairment in rats
Article
Year: 2021
Pages: 1
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Strictly regulated agonist-dependent activation of AMPA-R is the key characteristic of TAK-653 for robust synaptic responses and cognitive improvement
Article
Year: 2021
Pages: 1
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Isolation, characterization, anti-MRSA evaluation, and in-silico multi-target anti-microbial validations of actinomycin X
2
and actinomycin D produced by novel
Streptomyces smyrnaeus
UKAQ_23
Article
Year: 2021
Pages: 1
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Discovery of Taroxaz-104: The first potent antidote of SARS-CoV-2 VOC-202012/01 strain
Article
Year: 2021
Pages: 1
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DEELIG: A Deep Learning Approach to Predict Protein-Ligand Binding Affinity
Article
Year: 2021
Pages: 1
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In vitro efficacy of artemisinin-based treatments against SARS-CoV-2
Article
Year: 2021
Pages: 1
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A bivalent recombinant vaccine: a promising strategy against both SARS-CoV-2 variants and wild type of the virus
Article
Year: 2021
Pages: 1
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Can antidepressants unlock prescription of rimonabant in the fight against COVID-19?
Article
Year: 2021
Pages: 2
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Structure-based
in silico
approaches for drug discovery against
Mycobacterium tuberculosis
Article
Year: 2021
Pages: 12
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Identification of subtypes of anticancer peptides based on sequential features and physicochemical properties
Article
Year: 2021
Pages: 1
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Targeting oxidative stress in disease: promise and limitations of antioxidant therapy
Article
Year: 2021
Pages: 21
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YIV-906 potentiated anti-PD1 action against hepatocellular carcinoma by enhancing adaptive and innate immunity in the tumor microenvironment
Article
Year: 2021
Pages: 1
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NOD: a web server to predict
N
ew use of
O
ld
D
rugs to facilitate drug repurposing
Article
Year: 2021
Pages: 1
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The risk of major bleeding event in patients with chronic kidney disease on pentoxifylline treatment
Article
Year: 2021
Pages: 1
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The recombinant plant
Bauhinia bauhinioides
elastase inhibitor reduces rat thrombus without alterations in hemostatic parameters
Article
Year: 2021
Pages: 1
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Selection of safe artemisinin derivatives using a machine learning-based cardiotoxicity platform and in vitro and in vivo validation
Article
Year: 2021
Pages: 11
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Local application of
Usag-1
siRNA can promote tooth regeneration in
Runx2
-deficient mice
Article
Year: 2021
Pages: 1
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Rapid structure-based identification of potential SARS-CoV-2 main protease inhibitors
Article
Pages: 1
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All‐Atom Simulations and Free‐Energy Calculations of Antibodies Bound to the Spike Protein of SARS‐CoV‐2: The Binding Strength and Multivalent Hydrogen‐Bond Interactions
Article
Year: 2021
Pages: 1
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Editorial: Pharmacology of BPSD (Behavioral and Psychological Symptoms of Dementia)
Article
Year: 2021
Pages: 1
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Exploring the chemical space of protein–protein interaction inhibitors through machine learning
Article
Year: 2021
Pages: 1
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Stereoselective synthesis of a 4-⍺-glucoside of valienamine and its X-ray structure in complex with
Streptomyces coelicolor
GlgE1-V279S
Article
Year: 2021
Pages: 1
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There is no market for new antibiotics: this allows an open approach to research and development
Article
Year: 2021
Pages: 1
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Structures and Dynamics of Native-State Transmembrane Protein Targets and Bound Lipids
Article
Year: 2021
Pages: 1
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Zebrafish: An Attractive Model to Study
Staphylococcus aureus
Infection and Its Use as a Drug Discovery Tool
Article
Year: 2021
Pages: 1
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Molecular Human Targets of Bioactive Alkaloid-Type Compounds from
Tabernaemontana cymose
Jacq.
Article
Year: 2021
Pages: 1
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Patient-derived scaffolds as a drug-testing platform for endocrine therapies in breast cancer
Article
Year: 2021
Pages: 1
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Improving the Pharmacological Properties of Ciclopirox for Its Use in Congenital Erythropoietic Porphyria
Article
Year: 2021
Pages: 1
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Human Pluripotent Stem-Cell-Derived Models as a Missing Link in Drug Discovery and Development
Article
Year: 2021
Pages: 1
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A Structural Approach into Drug Discovery Based on Autophagy
Article
Year: 2021
Pages: 1
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In silico comparison of SARS-CoV-2 spike protein-ACE2 binding affinities across species and implications for virus origin
Article
Year: 2021
Pages: 1
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Author Correction: A therapeutic combination of two small molecule toxin inhibitors provides broad preclinical efficacy against viper snakebite
Article
Year: 2021
Pages: 1
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The c-Abl inhibitor, radotinib induces apoptosis in multiple myeloma cells via mitochondrial-dependent pathway
Article
Year: 2021
Pages: 1
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Attacking COVID-19 Progression Using Multi-Drug Therapy for Synergetic Target Engagement
Article
Year: 2021
Pages: 1
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New Quinone Antibiotics against Methicillin-Resistant
S. aureus
Article
Year: 2021
Pages: 1
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A Crystallographic Snapshot of SARS-CoV-2 Main Protease Maturation Process
Article
Year: 2021
Pages: 1
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Modeling the mature CNS: A predictive screening platform for neurodegenerative disease drug discovery
Article
Year: 2021
Pages: 1
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Polθ inhibitors elicit
BRCA
-gene synthetic lethality and target PARP inhibitor resistance
Article
Year: 2021
Pages: 1
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Genome-wide discovery of hidden genes mediating known drug-disease association using KDDANet
Article
Year: 2021
Pages: 1
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Artificial intelligence and machine learning‐aided drug discovery in central nervous system diseases: State‐of‐the‐arts and future directions
Article
Year: 2020
Pages: 47
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Pharmacologic targeting of Cdc42 GTPase by a small molecule Cdc42 activity-specific inhibitor prevents platelet activation and thrombosis
Article
Year: 2021
Pages: 1
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From Genome to Drugs: New Approaches in Antimicrobial Discovery
Article
Year: 2021
Pages: 1
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Evolving scenario of big data and Artificial Intelligence (AI) in drug discovery
Article
Year: 2021
Pages: 22
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CASTELO: clustered atom subtypes aided lead optimization—a combined machine learning and molecular modeling method
Article
Year: 2021
Pages: 1
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Partially Purified Leaf Fractions of
Azadirachta indica
Inhibit Trypanosome Alternative Oxidase and Exert Antitrypanosomal Effects on
Trypanosoma congolense
Article
Year: 2021
Pages: 10
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Drug target gene-based analyses of drug repositionability in rare and intractable diseases
Article
Year: 2021
Pages: 1
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Random forest classification for predicting lifespan-extending chemical compounds
Article
Year: 2021
Pages: 1
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Targeting mitochondrial reactive oxygen species-mediated oxidative stress attenuates nicotine-induced cardiac remodeling and dysfunction
Article
Year: 2021
Pages: 1
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A scaffolded approach to unearth potential antibacterial components from epicarp of Malaysian
Nephelium lappaceum
L.
Article
Year: 2021
Pages: 1
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Rhamnan sulphate from green algae
Monostroma nitidum
improves constipation with gut microbiome alteration in double-blind placebo-controlled trial
Article
Year: 2021
Pages: 1
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Strategic approach of multifaceted antibacterial mechanism of limonene traced in
Escherichia coli
Article
Year: 2021
Pages: 1
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Acetylcholinesterase and monoamine oxidase-B inhibitory activities by ellagic acid derivatives isolated from
Castanopsis cuspidata
var.
sieboldii
Article
Year: 2021
Pages: 1
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Radiation exposure induces cross-species temporal metabolic changes that are mitigated in mice by amifostine
Article
Year: 2021
Pages: 1
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Synergistic protective effects of lycopene and N-acetylcysteine against cisplatin-induced hepatorenal toxicity in rats
Article
Year: 2021
Pages: 1
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Alkaloids in Contemporary Drug Discovery to Meet Global Disease Needs
Article
Year: 2021
Pages: 1
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Antiviral Activity of Metabolites from Peruvian Plants against SARS-CoV-2: An In Silico Approach
Article
Year: 2021
Pages: 1
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Feature importance correlation from machine learning indicates functional relationships between proteins and similar compound binding characteristics
Article
Year: 2021
Pages: 1
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Insights into the molecular properties underlying antibacterial activity of prenylated (iso)flavonoids against MRSA
Article
Year: 2021
Pages: 1
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Dietary Flavonoids: Cardioprotective Potential with Antioxidant Effects and Their Pharmacokinetic, Toxicological and Therapeutic Concerns
Article
Year: 2021
Pages: 1
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In-vitro, in-vivo, and in-silico assessment of radical scavenging and cytotoxic activities of
Oliveria decumbens
essential oil and its main components
Article
Year: 2021
Pages: 1
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Uptake and release characteristics of serotonin hydrochloride by natural Cuban zeolite containing clinoptilolite and mordenite
Article
Year: 2021
Pages: 1
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Editorial: Recent Advances in G Protein-Coupled Receptor Signalling: Impact of Intracellular Location, Environment and Biased Agonism
Article
Year: 2021
Pages: 1
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Rational approach to drug discovery for human schistosomiasis
Article
Year: 2021
Pages: 8
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Structure-based redesigning of pentoxifylline analogs against selective phosphodiesterases to modulate sperm functional competence for assisted reproductive technologies
Article
Year: 2021
Pages: 1
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Taurine ameliorates thioacetamide induced liver fibrosis in rats via modulation of toll like receptor 4/nuclear factor kappa B signaling pathway
Article
Year: 2021
Pages: 1
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Transcriptomics-based drug repositioning pipeline identifies therapeutic candidates for COVID-19
Article
Year: 2021
Pages: 1
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The neural economics of brain aging
Article
Year: 2021
Pages: 1
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DNA-PK inhibitor peposertib enhances p53-dependent cytotoxicity of DNA double-strand break inducing therapy in acute leukemia
Article
Year: 2021
Pages: 1
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Spatiotemporal imaging and pharmacokinetics of fluorescent compounds in zebrafish eleuthero-embryos after different routes of administration
Article
Year: 2021
Pages: 1
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BING, a novel antimicrobial peptide isolated from Japanese medaka plasma, targets bacterial envelope stress response by suppressing
cpxR
expression
Article
Year: 2021
Pages: 1
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PB01 suppresses radio-resistance by regulating ATR signaling in human non-small-cell lung cancer cells
Article
Year: 2021
Pages: 1
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Bladder cancer therapy using a conformationally fluid tumoricidal peptide complex
Article
Year: 2021
Pages: 1
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Osmotically balanced, large unilamellar liposomes that enable sustained bupivacaine release for prolonged pain relief in in vivo rat models
Article
Year: 2021
Pages: 1
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PD-1 derived CA-170 is an oral immune checkpoint inhibitor that exhibits preclinical anti-tumor efficacy
Article
Year: 2021
Pages: 1
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Identification of anti‐Parkinson's Disease Lead Compounds from
Aspergillus ochraceus
Targeting Adenosin Receptors A
2A
Article
Year: 2021
Pages: 9
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A metabolic modeling approach reveals promising therapeutic targets and antiviral drugs to combat COVID-19
Article
Year: 2021
Pages: 1
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Combination treatment with U0126 and rt-PA prevents adverse effects of the delayed rt-PA treatment after acute ischemic stroke
Article
Year: 2021
Pages: 1
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Introduction to the EQIPD quality system
Article
Pages: 1
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Reprogramming of the Caseinolytic Protease by ADEP Antibiotics: Molecular Mechanism, Cellular Consequences, Therapeutic Potential
Article
Year: 2021
Pages: 1
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Aurora kinase A, a synthetic lethal target for precision cancer medicine
Article
Year: 2021
Pages: 13
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Anticancer drug discovery from Iranian
Chrysanthemum
cultivars through system pharmacology exploration and experimental validation
Article
Year: 2021
Pages: 1
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Generation of tetracycline-controllable CYP3A4-expressing Caco-2 cells by the piggyBac transposon system
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Year: 2021
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In vitro assessment and phase I randomized clinical trial of anfibatide a snake venom derived anti-thrombotic agent targeting human platelet GPIbα
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Inhibition of triple negative breast cancer metastasis and invasiveness by novel drugs that target epithelial to mesenchymal transition
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Year: 2021
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In silico identification of novel chemical compounds with antituberculosis activity for the inhibition of InhA and EthR proteins from Mycobacterium tuberculosis
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Transferrin-modified liposomes triggered with ultrasound to treat HeLa cells
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Is the oral microbiome a source to enhance mucosal immunity against infectious diseases?
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Association of the transthyretin variant V122I with polyneuropathy among individuals of African ancestry
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Maximizing the potential of aggressive mouse tumor models in preclinical drug testing
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Small Molecule Compounds Identified from Mixture-Based Library Inhibit Binding between
Plasmodium falciparum
Infected Erythrocytes and Endothelial Receptor ICAM-1
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Year: 2021
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Is Emodin with Anticancer Effects Completely Innocent? Two Sides of the Coin
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Suppression of Breast Cancer by Small Molecules That Block the Prolactin Receptor
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Pharmacological inhibition of noncanonical EED-EZH2 signaling overcomes chemoresistance in prostate cancer
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Year: 2021
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FragMAXapp
: crystallographic fragment-screening data-analysis and project-management system
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Year: 2021
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A Screening of the MMV Pandemic Response Box Reveals Epetraborole as A New Potent Inhibitor against
Mycobacterium abscessus
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Year: 2021
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When Good Kinases Go Rogue: GSK3, p38 MAPK and CDKs as Therapeutic Targets for Alzheimer’s and Huntington’s Disease
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VirtualFlow Ants—Ultra-Large Virtual Screenings with Artificial Intelligence Driven Docking Algorithm Based on Ant Colony Optimization
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Recent Applications of Deep Learning Methods on Evolution- and Contact-Based Protein Structure Prediction
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Small molecules in targeted cancer therapy: advances, challenges, and future perspectives
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Selective targeting of non-centrosomal AURKA functions through use of a targeted protein degradation tool
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Rationality over fashion and hype in drug design
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Schistosomiasis Drug Discovery in the Era of Automation and Artificial Intelligence
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Neuroprotective effect of selumetinib on acrolein-induced neurotoxicity
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New insights of phenolic compounds from optimized fruit extract of
Ficus auriculata
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Targeting
Mycobacterium tuberculosis
CoaBC through Chemical Inhibition of 4′-Phosphopantothenoyl-
l
-cysteine Synthetase (CoaB) Activity
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Year: 2021
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Development and validation of a high-throughput whole cell assay to investigate
Staphylococcus aureus
adhesion to host ligands
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Year: 2021
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Human pancreatic cancer cells under nutrient deprivation are vulnerable to redox system inhibition
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Year: 2021
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Co-crystal structures of HIV TAR RNA bound to lab-evolved proteins show key roles for arginine relevant to the design of cyclic peptide TAR inhibitors
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Year: 2021
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Long-term atomoxetine-oxybutynin combination use may be beneficial for the prevention of obstructive sleep apnea
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Year: 2021
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Evaluation of the anti-biofilm effect of poloxamer-based thermoreversible gel of silver nanoparticles as a potential medication for root canal therapy
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Discovery of New Potent anti-MERS CoV Fusion Inhibitors
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Year: 2021
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Pharmacologic modulation of 5-fluorouracil by folinic acid and high-dose pyridoxine for treatment of patients with digestive tract carcinomas
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Year: 2021
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Mutant p53s and chromosome 19 microRNA cluster overexpression regulate cancer testis antigen expression and cellular transformation in hepatocellular carcinoma
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Year: 2021
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Preclinical study to improve microbubble-mediated drug delivery in cancer using an ultrasonic probe with an interchangeable acoustic lens
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ELV-N32 and RvD6 isomer decrease pro-inflammatory cytokines, senescence programming, ACE2 and SARS-CoV-2-spike protein RBD binding in injured cornea
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An ACE2 Triple Decoy that neutralizes SARS-CoV-2 shows enhanced affinity for virus variants
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Progress on open chemoinformatic tools for expanding and exploring the chemical space
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Year: 2021
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Inhibition of MMP2-PEX by a novel ester of dihydroxy cinnamic and linoleic acid from the seagrass
Cymodocea serrulata
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Year: 2021
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Strategy for COVID-19 vaccination in India: the country with the second highest population and number of cases
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Daphnetin ameliorates acute lung injury in mice with severe acute pancreatitis by inhibiting the JAK2–STAT3 pathway
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Synthesis, photocatalytic and antidiabetic properties of ZnO/PVA nanoparticles
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Drug screening with zebrafish visual behavior identifies carvedilol as a potential treatment for an autosomal dominant form of retinitis pigmentosa
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Streamlined human antibody generation and optimization by exploiting designed immunoglobulin loci in a B cell line
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Year: 2020
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High fructose and streptozotocin induced diabetic impairments are mitigated by Indirubin-3-hydrazone via downregulation of PKR pathway in Wistar rats
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Synthesis of [
211
At]4-astato-L-phenylalanine by dihydroxyboryl-astatine substitution reaction in aqueous solution
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Fluorescent base analogues in gapmers enable stealth labeling of antisense oligonucleotide therapeutics
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Bardoxolone and bardoxolone methyl, two Nrf2 activators in clinical trials, inhibit SARS-CoV-2 replication and its 3C-like protease
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Berberine modulates hyper-inflammation in mouse macrophages stimulated with polyinosinic-polycytidylic acid via calcium-CHOP/STAT pathway
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Hydrogel with silver nanoparticles synthesized by
Mimosa tenuiflora
for second-degree burns treatment
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Ligand-Dependent Conformational Transitions in Molecular Dynamics Trajectories of GPCRs Revealed by a New Machine Learning Rare Event Detection Protocol
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Viral fibrotic scoring and drug screen based on MAPK activity uncovers EGFR as a key regulator of COVID-19 fibrosis
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A hybrid modeling approach for assessing mechanistic models of small molecule partitioning in vivo using a machine learning-integrated modeling platform
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A plant endophyte
Staphylococcus hominis
strain MBL_AB63 produces a novel lantibiotic, homicorcin and a position one variant
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PPI Modulators of E6 as Potential Targeted Therapeutics for Cervical Cancer: Progress and Challenges in Targeting E6
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HDAC6 inhibitors sensitize non-mesenchymal triple-negative breast cancer cells to cysteine deprivation
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Preclinical and clinical characterization of the RORγt inhibitor JNJ-61803534
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Novel human neutralizing mAbs specific for Spike-RBD of SARS-CoV-2
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Structural Requirements for Dihydrobenzoxazepinone Anthelmintics: Actions against Medically Important and Model Parasites:
Trichuris muris
,
Brugia malayi
,
Heligmosomoides polygyrus
, and
Schistosoma mansoni
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Year: 2021
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Opportunities and Challenges in Developing a
Cryptosporidium
Controlled Human Infection Model for Testing Antiparasitic Agents
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Multiple unbiased approaches identify oxidosqualene cyclase as the molecular target of a promising anti-leishmanial
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Drug Target Identification with Machine Learning: How to Choose Negative Examples
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Xmrks the Spot: Fish Models for Investigating Epidermal Growth Factor Receptor Signaling in Cancer Research
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Deciphering the scopolamine challenge rat model by preclinical functional MRI
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Ubiquitination Regulators Discovered by Virtual Screening for the Treatment of Cancer
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Year: 2021
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High-throughput screening identifies a novel natural product-inspired scaffold capable of inhibiting
Clostridioides difficile
in vitro
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Year: 2021
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Identification of hepatic fibrosis inhibitors through morphometry analysis of a hepatic multicellular spheroids model
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Investigating auranofin for the treatment of infected diabetic pressure ulcers in mice and dermal toxicity in pigs
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Library of Selenocyanate and Diselenide Derivatives as In Vivo Antichagasic Compounds Targeting
Trypanosoma cruzi
Mitochondrion
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Year: 2021
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Ubiquitination, Biotech Startups, and the Future of TRIM Family Proteins: A TRIM-Endous Opportunity
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Integrative web-based analysis of omics data for study of drugs against SARS-CoV-2
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A novel synthetic microtubule inhibitor exerts antiproliferative effects in multidrug resistant cancer cells and cancer stem cells
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Editorial: Going the Distance: Enabling 3D Cell Culture Systems for Biomedical Research and Drug Treatment
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Computational study of the therapeutic potentials of a new series of imidazole derivatives against SARS-CoV-2
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Rational design of innate defense regulator peptides as tumor vaccine adjuvants
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Whole transcriptome RNA-seq reveals key regulatory factors involved in type 2 diabetes pathology in peripheral fat of Asian Indians
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A super-potent tetramerized ACE2 protein displays enhanced neutralization of SARS-CoV-2 virus infection
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Arylmethylene hydrazine derivatives containing 1,3-dimethylbarbituric moiety as novel urease inhibitors
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Towards water-soluble [60]fullerenes for the delivery of siRNA in a prostate cancer model
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Implementing a method for engineering multivalency to substantially enhance binding of clinical trial anti-SARS-CoV-2 antibodies to wildtype spike and variants of concern proteins
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Functional and structural characterization of a two-MAb cocktail for delayed treatment of enterovirus D68 infections
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Modulating Target Protein Biology Through the Re-mapping of Conformational Distributions Using Small Molecules
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Identification of targets of JS-K against HBV-positive human hepatocellular carcinoma HepG2.2.15 cells with iTRAQ proteomics
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Cisplatin and phenanthriplatin modulate long-noncoding RNA expression in A549 and IMR90 cells revealing regulation of microRNAs, Wnt/β-catenin and TGF-β signaling
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Outer membrane and phospholipid composition of the target membrane affect the antimicrobial potential of first- and second-generation lipophosphonoxins
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Rational Design of Peptide-Based Inhibitors Disrupting Protein-Protein Interactions
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Kinase drug discovery 20 years after imatinib: progress and future directions
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Discovery of (
E
)-
N
-(4-cyanobenzylidene)- 6-fluoro- 3-hydroxypyrazine-2 -carboxamide (cyanorona-20): the first potent and specific anti-COVID-19 drug
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Year: 2021
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A Soluble Epoxide Hydrolase Inhibitor, 1-trifluoromethoxyphenyl-3-(1-propionylpiperidin-4-yl) Urea, Ameliorates Experimental Autoimmune Encephalomyelitis
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Small Molecules of Marine Origin as Potential Anti-Glioma Agents
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Advances in Applying Computer-Aided Drug Design for Neurodegenerative Diseases
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Medicinal Plants with Anti-Leukemic Effects: A Review
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Year: 2021
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Recent Advances in Discovery of Lead Structures from Microbial Natural Products: Genomics- and Metabolomics-Guided Acceleration
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A Novel Method to Predict Drug-Target Interactions Based on Large-Scale Graph Representation Learning
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Tubulin Inhibitors: A Chemoinformatic Analysis Using Cell-Based Data
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Year: 2021
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Peptides to Tackle Leishmaniasis: Current Status and Future Directions
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Year: 2021
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PyPLIF HIPPOS-Assisted Prediction of Molecular Determinants of Ligand Binding to Receptors
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Synthesis of New Triazolopyrazine Antimalarial Compounds
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Year: 2021
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Phytochemicals from Ajwa dates pulp extract induce apoptosis in human triple-negative breast cancer by inhibiting AKT/mTOR pathway and modulating Bcl-2 family proteins
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Year: 2021
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Adalimumab biosimilars, ABP501 and SB5, are equally effective and safe as adalimumab originator
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Year: 2021
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Drug repurposing for ligand-induced rearrangement of Sirt2 active site-based inhibitors via molecular modeling and quantum mechanics calculations
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Year: 2021
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Repurposing ketoconazole as an exosome directed adjunct to sunitinib in treating renal cell carcinoma
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Year: 2021
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Process optimization for the supercritical carbondioxide extraction of lycopene from ripe grapefruit (
Citrus paradisi
) endocarp
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Year: 2021
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Development of P301S tau seeded organotypic hippocampal slice cultures to study potential therapeutics
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Year: 2021
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Discovery and characterization of small-molecule inhibitors of NLRP3 and NLRC4 inflammasomes
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Year: 2021
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Highlighting membrane protein structure and function: A celebration of the Protein Data Bank
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Year: 2021
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Edelfosine nanoemulsions inhibit tumor growth of triple negative breast cancer in zebrafish xenograft model
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Year: 2021
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d
-Cystine di(m)ethyl ester reverses the deleterious effects of morphine on ventilation and arterial blood gas chemistry while promoting antinociception
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Year: 2021
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Applications of Virtual Screening in Bioprospecting: Facts, Shifts, and Perspectives to Explore the Chemo-Structural Diversity of Natural Products
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Selective and noncovalent targeting of RAS mutants for inhibition and degradation
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Year: 2021
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Acute toxicity analysis of an inhibitor of BCL2, Disarib, in rats
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Year: 2021
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Antiplasmodial activity of the natural product compounds alstonine and himbeline
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Year: 2021
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N
-Demethylsinomenine, an active metabolite of sinomenine, attenuates chronic neuropathic and inflammatory pain in mice
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Year: 2021
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SMMPPI: a machine learning-based approach for prediction of modulators of protein–protein interactions and its application for identification of novel inhibitors for RBD:hACE2 interactions in SARS-CoV-2
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Year: 2021
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Editorial: New Approaches Against Drug-Resistant
M. tuberculosis
Article
Year: 2021
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Central administration of afzelin extracted from
Ribes fasciculatum
improves cognitive and memory function in a mouse model of dementia
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Year: 2021
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Discovery of a novel RORγ antagonist with skin-restricted exposure for topical treatment of mild to moderate psoriasis
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Year: 2021
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Potent synthetic and endogenous ligands for the adopted orphan nuclear receptor Nurr1
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Year: 2021
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Human WRN is an intrinsic inhibitor of progerin, abnormal splicing product of lamin A
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Year: 2021
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Cytotoxic, analgesic and anti-inflammatory activity of colchicine and its C-10 sulfur containing derivatives
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Year: 2021
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Editorial: Molecular Dynamics and Machine Learning in Drug Discovery
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Year: 2021
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P2X3 Receptor Ligands: Structural Features and Potential Therapeutic Applications
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Year: 2021
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A novel cystathionine γ-lyase inhibitor, I194496, inhibits the growth and metastasis of human TNBC via downregulating multiple signaling pathways
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Year: 2021
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Artificially Induced Pluripotent Stem Cell-Derived Whole-Brain Organoid for Modelling the Pathophysiology of Metachromatic Leukodystrophy and Drug Repurposing
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Year: 2021
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RHO to the DOCK for GDP disembarking: Structural insights into the DOCK GTPase nucleotide exchange factors
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Year: 2021
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Ligand-Receptor Interactions and Machine Learning in GCGR and GLP-1R Drug Discovery
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Year: 2021
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Facile Synthesis and In Vitro Activity of
N
-Substituted 1,2-Benzisothiazol-3(2
H
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Year: 2021
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A Network Medicine Approach for Drug Repurposing in Duchenne Muscular Dystrophy
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Year: 2021
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Downregulating carnitine palmitoyl transferase 1 affects disease progression in the SOD1 G93A mouse model of ALS
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Year: 2021
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Targeting protein-protein interaction interfaces in COVID-19 drug discovery
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Year: 2021
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GPCR_LigandClassify.py; a rigorous machine learning classifier for GPCR targeting compounds
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Year: 2021
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SANCDB: an update on South African natural compounds and their readily available analogs
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Year: 2021
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Temporal activation of WNT/β-catenin signaling is sufficient to inhibit SOX10 expression and block melanoma growth
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Year: 2020
Pages: 23
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Intrinsically Disordered Proteins as Regulators of Transient Biological Processes and as Untapped Drug Targets
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Year: 2021
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Editorial: Understanding Protein Dynamics, Binding and Allostery for Drug Design
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Year: 2021
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FoldAffinity: binding affinities from nDSF experiments
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Year: 2021
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